ALLEGATO 1. - SOMMARIO DI ALCUNE CARATTERISTICHE DEI FARMACI ANTIRETROVIRALI DISPONIBILI 1.A) Inibitori della transcriptasi inversa _____________________________________________________________________ | |Zidovudina|Didanosina|Zalcitabina|Lamivudina|Stavudina| |____________|__________|__________|___________|__________|_________| |Abbrevazione|AZT |ddl |ddC |3TC |d4T | |____________|__________|__________|___________|__________|_________| |Nome |Retrovir |Videx |Hivid |Epivir |Zerit | |commerciale | | | | | | |____________|__________|__________|___________|__________|_________| |Posologia | 2x250 mg | 2x200 mg | 3x0.75 mg | 2x150 mg | 2x40 mg | |abituale | 3x200 mg | | | | | |____________|__________|__________|___________|__________|_________| |Effetti |Anemia, |Diarrea, |Neuropatia,|Cefalea, |Neuropa- | |collaterali |neutrope- |pancreati-|ulcere |nausea |tie | |piu' |nia |te |orali | | | |frequenti | | | | | | |____________|__________|__________|___________|__________|_________| 1.B) Inibitori della proteasi _____________________________________________________________________ | |Indinavir |Ritonavir |Saquinavir | |_______________|________________|_________________|________________| |Nome |Crixivan |Norvir |Invirase | |commerciale | | | | |_______________|________________|_________________|________________| |Posologia | 3x800 mg | 2x600 mg | 3x600 mg, | | | | | dopo i pasti | |_______________|________________|_________________|________________| |Effetti |Iperbilirubine- |Nausea, diarrea, |Disturbi | |collaterali |mia nefrolitiasi|neuropatia |gastrointestina-| |piu' frequenti | |circumorale e |li | | | |periferica | | |_______________|________________|_________________|________________|